SCHEMBL4581069

SCHEMBL4581069

O=C1NCCN(c2ccnc(Nc3cccc([N+](=O)[O-])c3)n2)C1c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.49
BCR P11274 3/20 0.49
PRKCA P17252 3/20 0.49
EGFR P00533 2/20 0.46
SRC P12931 1/20 0.46
CDK2 P24941 8/20 0.45
CDK4 P11802 6/20 0.44
GSK3B P49841 2/20 0.43
SLC2A1 P11166 1/20 0.43
CCNT1 O60563 3/20 0.43
CDK9 P50750 3/20 0.43
CCNA2 P20248 3/20 0.42
CDK5 Q00535 2/20 0.42
CDK5R1 Q15078 2/20 0.42
PTK6 Q13882 1/20 0.42
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CDK7 P50613 2/20 0.42
CCNH P51946 2/20 0.42
AURKA O14965 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4582376 0.87 KDR (0.43) ABL1PRKCAEGFRCDK2CDK1
SCHEMBL4581040 0.85 KDR (0.51) ABL1BCREGFRSRCCDK2
SCHEMBL4582327 0.85 HDAC1 (0.47) CDK2CDK4GSK3BCDK9CDK5
SCHEMBL4580811 0.85 KDR (0.51) ABL1BCRPRKCACDK2CDK4
SCHEMBL4581942 0.84 IKBKB (0.46) CDK2CDK4GSK3B
SCHEMBL4579436 0.83 FLT1 (0.52) EGFRCDK2GSK3BCDK5CDK1
SCHEMBL4580715 0.81 PIK3CA (0.52) ABL1CDK2CDK4GSK3BCDK9
SCHEMBL4580865 0.80 MAPK14 (0.42) EGFRGSK3BALDH1A1KMT2ASMN1; SMN2
SCHEMBL4580975 0.80 IKBKB (0.41) CDK2GSK3BPLK1ALDH1A1KMT2A
SCHEMBL4581955 0.79 IKBKB (0.42) CDK2CDK4GSK3BCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US claimed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US claimed
US-7323464-B2 Pyridine and pyrimidine derivatives CELLTECH R&D LIMITED (GB) 2008-01-29 US disclosed
US-20050080258-A1 Pyridine and pyrimidine derivatives GENTEX CORPORATION 2005-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080258-A1 Pyridine and pyrimidine derivatives ROR1, MAPK1, IRAK1 ABL1 32/4885BCR 63/4885PRKCA 1303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.