SCHEMBL458234

SCHEMBL458234

O=C(OCc1ccccc1)N1CCC(CCOc2cnc(Cl)nc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 11/20 0.55
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
CYP2D6 P10635 4/20 0.53
CYP2C9 P11712 4/20 0.53
CYP3A4 P08684 3/20 0.53
FAAH O00519 1/20 0.53
CYP2C19 P33261 1/20 0.52
CHRM4 P08173 2/20 0.52
TEAD1 P28347 1/20 0.49
TEAD3 Q99594 1/20 0.49
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458097 0.89 GRIN2B (0.57) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL20590855 0.85 GRIN2B (0.53) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL25208669 0.84 SMN1; SMN2 (0.57) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL20207185 0.83 SMN1; SMN2 (0.57) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL5231915 0.83 GRIN2B (0.57) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL457685 0.80 GRIN2B (0.50) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL15140566 0.80 SMN1; SMN2 (0.72) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL470480 0.80 SMN1; SMN2 (0.53) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL9411411 0.79 SMN1; SMN2 (0.64) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6
SCHEMBL8765520 0.78 SMN1; SMN2 (0.62) GRIN2BSMN1; SMN2NPC1RAB9ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011147951-A1 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS PROSIDION LIMITED (GB) 2011-12-01 WO disclosed