SCHEMBL458420

SCHEMBL458420

C1=C\N=N/N=N\N=C/1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2494 1.00
Hydrochloric Acid SCHEMBL17303190 0.97
SCHEMBL29138664 0.85
Cadaverine Tartrate SCHEMBL7865850 0.78 TSHR (0.39)
Cadaverine Tartrate SCHEMBL9163185 0.77 TSHR (0.37)
Hydrochloric Acid SCHEMBL5490018 0.77
SCHEMBL29771444 0.75
SCHEMBL84535 0.71
SCHEMBL84537 0.71
SCHEMBL84536 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1130 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4100010-B1 NITROXIDE COMPOUNDS FOR USE IN THE TREATMENT OF OPIOID-INDUCED RESPIRATORY DEPRESSION (OIRD) UNIV CASE WESTERN RESERVE (US) 2026-01-07 EP claimed
EP-3180349-B1 LYMPH DIRECTING PRODRUGS AND THERAPEUTIC USES THEREOF UNIV MONASH (AU) 2025-03-12 EP claimed
EP-3441087-B1 METHODS OF TREATING CHRONIC PAIN TEVA PHARMACEUTICALS INT GMBH (CH) 2025-02-19 EP claimed
EP-3706762-B1 N4-HYDROXYCYTIDINE DERIVATIVE AND ANTI-VIRAL USES RELATED THERETO UNIV EMORY (US) 2024-10-16 EP claimed
EP-3863708-B1 MIXED IONIC CONDUCTORS AND CORRESPONDING DEVICES, SYSTEMS AND METHODS OF MAKING BATTELLE MEMORIAL INSTITUTE (US) 2024-09-11 EP claimed
EP-3768679-B1 BIASED POTENT OPIOID-LIKE AGONISTS AS IMPROVED MEDICATIONS TO TREAT CHRONIC AND ACUTE PAIN AND METHODS OF USING THE SAME US HEALTH (US) 2024-06-26 EP claimed
EP-1962797-B2 POWDER COMPOSITIONS FOR INHALATION JAGOTEC AG (CH) 2024-05-29 EP claimed
EP-3682872-B1 LIQUISOFT CAPSULES PATHEON SOFTGELS INC (US) 2024-01-03 EP claimed
EP-0300806-B1 Opioid analgesic liposomal delivery-release system VESTAR INC (US) 1994-09-07 EP claimed
EP-0367746-B1 Sustained release drug-resin complexes RICHARDSON VICKS INC (US) 1994-02-02 EP claimed
EP-0441833-B1 DOSAGE FORM HAVING REDUCED ABUSE POTENTIAL ALZA CORPORATION (US) 1993-09-08 EP claimed
WO-1993002707-A1 NEW ANTI-DIARRHEIC AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-02-18 WO claimed
EP-0375689-B1 A PHARMACEUTICAL COMPOSITION ADAPTED FOR TRANSDERMAL DELIVERY OF AN OPOID DRUG. WARNER-LAMBERT COMPANY (US) 1992-08-12 EP claimed
EP-0287469-B1 MIXTURE CONTAINING AS THE ACTIVE PRINCIPLES A CENTRAL ANALGESIC AND FORSKOLIN ROUSSEL-UCLAF (FR) 1992-07-08 EP claimed
EP-0108017-B1 MIXTURE COMPRISING A CENTRAL ANALGESIC AND VITAMIN B12, OR ONE OF ITS ANALOGS, AS ACTIVE PRINCIPLES ROUSSEL-UCLAF (FR) 1986-12-10 EP claimed
EP-0046270-B1 NOVEL DERIVATIVES OF BIO-AFFECTING PHENOLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM INTERx RESEARCH CORPORATION (US) 1986-05-21 EP claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
EP-0036145-B1 AN ORALLY ADMINISTERED DRUG FORM COMPRISING A POLAR BIOACTIVE AGENT AND AN ADJUVANT INTERx RESEARCH CORPORATION (US) 1985-05-29 EP claimed