SCHEMBL4585760

SCHEMBL4585760

OC1CCC(n2ccnc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
HRH1 P35367 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP19A1 P11511 3/20 0.35
F10 P00742 1/20 0.33
CYP17A1 P05093 2/20 0.33
CYP2B6 P20813 1/20 0.32
HCAR1 Q9BXC0 1/20 0.31
CPB2 Q96IY4 1/20 0.31
CD38 P28907 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
NFKB1 P19838 1/20 0.30
QPCT Q16769 1/20 0.30
HSD17B10 Q99714 1/20 0.30
QPCTL Q9NXS2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809415 1.00 CYP3A4 (0.35) CYP3A4CYP2D6HRH1KCNH2CYP19A1
SCHEMBL945421 0.89
Hydrochloric Acid SCHEMBL28498519 0.87 CYP19A1 (0.39) CYP3A4CYP2D6HRH1KCNH2CYP19A1
Ammonia Solution, Strong SCHEMBL28860953 0.87
SCHEMBL21827988 0.81 CYP19A1 (0.36) CYP19A1CYP17A1NFKB1QPCTHSD17B10
SCHEMBL21827989 0.81 CYP19A1 (0.36) CYP19A1CYP17A1NFKB1QPCTHSD17B10
SCHEMBL10068593 0.80
SCHEMBL4872099 0.80 CYP2B6 (0.44) CYP3A4CYP2D6HRH1KCNH2CYP19A1
SCHEMBL18055795 0.79 CYP19A1 (0.35) CYP19A1CYP17A1NFKB1QPCTHSD17B10
SCHEMBL31058221 0.79 CYP3A4 (0.35) CYP3A4CYP2D6HRH1KCNH2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0961618-A4 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-07-17 EP claimed
EP-0961618-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-08 EP claimed
WO-1998025619-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-06-18 WO claimed
WO-2023215991-A1 DNA-PK INHIBITOR COMPOUNDS AND USES THEREOF adMare Therapeutics Society (CA) 2023-11-16 WO disclosed
EP-1583535-A4 METHODS FOR TREATING DIABETES SCIOS INC (US) 2008-03-19 EP disclosed
EP-1583535-A2 METHODS FOR TREATING DIABETES SCIOS INC. (US) 2005-10-12 EP disclosed
WO-2004053107-A2 METHODS FOR TREATING DIABETES SCIOS INC. (US) 2004-06-24 WO disclosed
EP-0961618-A4 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-07-17 EP disclosed
EP-0961618-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-08 EP disclosed
WO-1998025619-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-06-18 WO disclosed