SCHEMBL4586249

SCHEMBL4586249

O=C(N[C@H](Cc1ccc2[nH]nnc2c1)C(=O)[N+]1(C2CCNCC2)CCCCC1)N1CCC(N2Cc3ccccc3NC2=O)CC1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.59
CYP3A4 P08684 16/20 0.59
CALCA P06881 1/20 0.48
RAMP1 O60894 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30231179 0.83 CALCRL (0.83) CALCRLCYP3A4
SCHEMBL13081467 0.83 CALCRL (0.83) CALCRLCYP3A4
SCHEMBL3764531 0.83 CALCRL (0.83) CALCRLCYP3A4
SCHEMBL3588012 0.83 CALCRL (0.63) CALCRLCYP3A4CALCA
SCHEMBL3588008 0.83 CALCRL (0.63) CALCRLCYP3A4CALCA
SCHEMBL30231279 0.83 CALCRL (0.63) CALCRLCYP3A4CALCA
SCHEMBL14526916 0.80 CALCRL (0.60) CALCRLCYP3A4CALCARAMP1
SCHEMBL13081132 0.80 CALCRL (0.58) CALCRLCYP3A4CALCA
SCHEMBL14526922 0.80 CALCRL (0.64) CALCRLCYP3A4RAMP1
SCHEMBL14526919 0.79 CALCRL (0.65) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689493-A4 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-04-23 EP disclosed
EP-1689493-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS Bristol-Myers Squibb Pharma Company (US) 2006-08-16 EP disclosed
WO-2005065779-A1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-21 WO disclosed