SCHEMBL4589190

SCHEMBL4589190

NC1CN(CC(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.46
HRH1 P35367 2/20 0.43
ALDH1A1 P00352 1/20 0.42
KCNA3 P22001 1/20 0.42
HTR2A P28223 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
GRIN2B Q13224 1/20 0.40
KDM4E B2RXH2 1/20 0.38
GRM2 Q14416 1/20 0.38
GRM3 Q14832 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079642 0.85 KCNA3 (0.53) CYP2D6HRH1ALDH1A1KCNA3SIGMAR1
SCHEMBL6079635 0.85 KCNA3 (0.53) CYP2D6HRH1ALDH1A1KCNA3SIGMAR1
SCHEMBL6080224 0.85 KCNA3 (0.53) CYP2D6HRH1ALDH1A1KCNA3SIGMAR1
SCHEMBL9595556 0.81 KCNA3 (0.47) CYP2D6ALDH1A1KCNA3SIGMAR1KDM4E
SCHEMBL10748973 0.80 KCNA3 (0.50) CYP2D6ALDH1A1KCNA3SIGMAR1GRIN2B
SCHEMBL28338145 0.77 KMT2A (0.57) ALDH1A1KCNA3KDM4EGRM2GRM3
Hydrochloric Acid SCHEMBL28637829 0.75 KMT2A (0.46) CYP2D6ALDH1A1KCNA3GRM2GRM3
SCHEMBL6079142 0.73 KCNA3 (0.64) CYP2D6KCNA3SIGMAR1
SCHEMBL6079135 0.73 KCNA3 (0.64) CYP2D6KCNA3SIGMAR1
SCHEMBL6079873 0.73 KCNA3 (0.64) CYP2D6KCNA3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060767-A2 MACROCYCLIC BENZOFUSED PYRIMIDINE DERIVATIVES ABBOTT LABORATORIES (US) 2008-05-22 WO disclosed