SCHEMBL4590676

SCHEMBL4590676

Clc1ccc(-n2ccc3cc(OCCCCCCBr)ccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.44
MCHR1 Q99705 2/20 0.39
KCNH2 Q12809 1/20 0.39
MCL1 Q07820 2/20 0.38
CYP19A1 P11511 1/20 0.38
HRH3 Q9Y5N1 6/20 0.36
ROCK2 O75116 1/20 0.36
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590763 0.99 BIRC5 (0.46) BIRC5MCHR1KCNH2MCL1CYP19A1
SCHEMBL5736518 0.88 KCNH2 (0.47) MCHR1KCNH2HRH3
SCHEMBL5736911 0.88 KCNH2 (0.47) MCHR1KCNH2HRH3
SCHEMBL5737170 0.87 SLC6A2 (0.44) KCNH2
SCHEMBL5735387 0.87 FGFR1 (0.46)
SCHEMBL5736908 0.86 KCNH2 (0.48) MCHR1KCNH2HRH3
SCHEMBL5735248 0.82 KCNH2 (0.49) MCHR1KCNH2HRH3
SCHEMBL5736008 0.78 BIRC5 (0.40) BIRC5KCNH2CYP19A1
SCHEMBL4591158 0.78 HRH3 (0.46) MCHR1KCNH2HRH3
SCHEMBL6561694 0.77 FGFR1 (0.47) BIRC5MCHR1KCNH2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107322-A1 INDOLE, BENZIMIDAZOLE OR BENZOTRIAZOLE DERIVATIVES INCLUDING A PIPERIDINE OR PIPERAZINE CORE AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed