SCHEMBL459221

SCHEMBL459221

Fc1cncc(-n2cnc3ccccc32)c1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.57
FGFR1 P11362 7/20 0.51
CYP17A1 P05093 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30423052 0.89 HTT (0.67) HTTFGFR1CYP17A1
SCHEMBL27241688 0.83 HTT (0.65) HTTFGFR1
SCHEMBL29949277 0.81 HTT (0.57) HTTFGFR1CYP17A1
SCHEMBL28848729 0.81 FGFR1 (0.68) HTTFGFR1
SCHEMBL22554097 0.81 HTT (0.57) HTTFGFR1CYP17A1
SCHEMBL30366915 0.81 HTT (0.57) HTTFGFR1CYP17A1
SCHEMBL29949104 0.81 FGFR1 (0.68) HTTFGFR1
SCHEMBL28848737 0.81 HTT (0.57) HTTFGFR1CYP17A1
SCHEMBL29898319 0.81 FGFR1 (0.67) HTTFGFR1
SCHEMBL27728245 0.81 FGFR1 (0.67) HTTFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed