SCHEMBL4592826

SCHEMBL4592826

CCc1c(N)cc(Cl)c(CC)c1NC(=O)N(c1ccc(OC)cc1)C(C)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
UTS2R Q9UKP6 13/20 0.43
CNR2 P34972 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
BCL2A1 Q16548 2/20 0.36
BID P55957 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592825 1.00 UTS2R (0.43) UTS2RCNR2FNTAFNTBBCL2A1
SCHEMBL5049344 0.95 MEN1 (0.39) UTS2RALDH1A1TAS1R3TAS1R1
SCHEMBL5050236 0.95 MEN1 (0.39) UTS2RALDH1A1TAS1R3TAS1R1
SCHEMBL5049341 0.95 MEN1 (0.39) UTS2RALDH1A1TAS1R3TAS1R1
SCHEMBL4592817 0.93 UTS2R (0.38) UTS2RBCL2A1BID
SCHEMBL4592820 0.93 UTS2R (0.38) UTS2RBCL2A1BID
SCHEMBL4592462 0.91 UTS2R (0.37) UTS2RBCL2A1BID
SCHEMBL4592463 0.91 UTS2R (0.37) UTS2RBCL2A1BID
SCHEMBL4592260 0.90 UTS2R (0.36) UTS2RBCL2A1BID
SCHEMBL4592262 0.90 UTS2R (0.36) UTS2RBCL2A1BID

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8071810-B2 3-(3-Amino-2,6-diisopropyl-phenyl)-1-(4-isopropyl-phenyl)-1-(4-methoxy-benzyl)-urea; autoimmune disorders; inflammation JERINI AG (DE) 2011-12-06 US claimed
US-20080220003-A1 C5a Receptor Antagonists JERINI AG (DE) 2008-09-11 US claimed
EP-1885691-A1 C5A RECEPTOR ANTAGONISTS Jerini AG (DE) 2008-02-13 EP claimed
WO-2006128670-A1 C5A RECEPTOR ANTAGONISTS JERINI AG (DE) 2006-12-07 WO claimed
US-8071810-B2 3-(3-Amino-2,6-diisopropyl-phenyl)-1-(4-isopropyl-phenyl)-1-(4-methoxy-benzyl)-urea; autoimmune disorders; inflammation JERINI AG (DE) 2011-12-06 US disclosed
US-20080220003-A1 C5a Receptor Antagonists JERINI AG (DE) 2008-09-11 US disclosed
EP-1885691-A1 C5A RECEPTOR ANTAGONISTS Jerini AG (DE) 2008-02-13 EP disclosed
WO-2006128670-A1 C5A RECEPTOR ANTAGONISTS JERINI AG (DE) 2006-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080220003-A1 C5a Receptor Antagonists C3AR1, C5AR2, C5AR1 UTS2R 206/4885CNR2 14/4885FNTA 2736/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.