SCHEMBL4593128

SCHEMBL4593128

O=C(O)c1ccc(Nc2ncnc3sccc23)c(OC2CCOC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
EGFR P00533 11/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ERBB2 P04626 1/20 0.42
KCNH2 Q12809 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794752 0.92 MEN1 (0.47) ALDH1A1GAAMEN1KMT2AEGFR
SCHEMBL3799137 0.91 NPC1 (0.54) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL3794854 0.91 MEN1 (0.48) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL3796447 0.85 MKNK2 (0.54) MEN1KMT2AEGFRRAB9AMKNK1
SCHEMBL4594135 0.83 MKNK2 (0.47) GAAEGFRMAPTMKNK1MKNK2
SCHEMBL3798528 0.83 MEN1 (0.49) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL3794289 0.83 MEN1 (0.49) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL3794275 0.82 EGFR (0.48) EGFRERBB2KCNH2
SCHEMBL13434909 0.81 MKNK1 (0.42) EGFRERBB2KCNH2PDE4APDE4B
SCHEMBL3795348 0.81 MEN1 (0.48) MEN1KMT2AEGFRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899353-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DeveloGen Aktiengesellschaft (DE) 2008-03-19 EP claimed
WO-2006136402-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DEVELOGEN AKTIENGESELLSCHAFT (DE) 2006-12-28 WO claimed