SCHEMBL4593652

SCHEMBL4593652

COc1ccc(C(C(N)=O)C(N)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.57
CA2 P00918 5/20 0.57
PARP10 Q53GL7 2/20 0.57
PARP1 P09874 1/20 0.57
PARP2 Q9UGN5 1/20 0.57
PARP4 Q9UKK3 1/20 0.57
RAB9A P51151 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
ALOX5 P09917 2/20 0.53
NPC1 O15118 1/20 0.53
MAPT P10636 1/20 0.53
PAX8 Q06710 1/20 0.53
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CA12 O43570 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10583234 0.90 PARP10 (0.52) CA1CA2PARP10PARP1PARP2
SCHEMBL11210093 0.90 NPC1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL4507705 0.85 CA1 (0.55) CA1CA2PARP10PARP1PARP2
SCHEMBL1115061 0.83 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL2055565 0.83 EPHX1 (0.55) CA1CA2PARP10PARP1PARP2
SCHEMBL2879870 0.83 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL2370549 0.83 EPHX1 (0.55) CA1CA2PARP10PARP1PARP2
SCHEMBL1354444 0.83 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL15517793 0.83 CA1 (0.53) CA1CA2PARP10PARP1PARP2
SCHEMBL5528055 0.83 CA1 (0.53) CA1CA2PARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104302287-B Indolin-2-one derivatives as protein kinase inhibitors 安基生技新药股份有限公司 2017-12-26 CN disclosed
EP-1957498-A2 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING MethylGene Inc. (CA) 2008-08-20 EP disclosed
WO-2008041053-A2 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE, INC. (CA) 2008-04-10 WO disclosed