SCHEMBL4596672

SCHEMBL4596672

Cc1nn(-c2ccccc2)c2nc(C3CN(C(=O)NCCc4ccc(F)cc4)C3)[nH]c(=O)c12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KHK P50053 6/20 0.54
TP53 P04637 1/20 0.45
NR3C1 P04150 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
CCNE1 P24864 4/20 0.44
CDK2 P24941 4/20 0.44
CDK1 P06493 2/20 0.44
CCNB1 P14635 2/20 0.44
MAPT P10636 2/20 0.43
TNF P01375 1/20 0.42
ATM Q13315 1/20 0.42
NOD2 Q9HC29 1/20 0.42
NOD1 Q9Y239 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4512852 0.92 KHK (0.55) KHKTP53ALDH1A1HPGDHTT
SCHEMBL4521006 0.86 KHK (0.58) KHKNR3C1ALDH1A1HPGDHTT
SCHEMBL4522989 0.86 KHK (0.60) KHKTP53ALDH1A1HPGDHTT
SCHEMBL4511884 0.83 KHK (0.54) KHKALDH1A1HPGDHTTCCNE1
SCHEMBL4505301 0.82 KHK (0.54) KHKTP53NR3C1HPGDCCNE1
SCHEMBL4522433 0.82 KHK (0.53) KHKTP53NR3C1CCNE1CDK2
SCHEMBL4507115 0.81 KHK (0.63) KHKNR3C1ALDH1A1HPGDHTT
SCHEMBL13865810 0.79 KHK (0.51) KHKNR3C1ALDH1A1HPGDHTT
SCHEMBL4502264 0.78 KHK (0.59) KHKALDH1A1HPGDHTTCCNE1
SCHEMBL4500604 0.78 KHK (0.48) KHKTP53ALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055959-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-05-15 WO disclosed