SCHEMBL4596731

SCHEMBL4596731

C[C@@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)C[C@H](C)[N+]1(C(=O)[O-])C(C)(C)C

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MLNR O43193 19/20 0.69
CYP3A4 P08684 7/20 0.69
CYP2D6 P10635 2/20 0.52
KCNH2 Q12809 1/20 0.52
GHSR Q92847 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596914 0.87 MLNR (0.71) MLNRCYP3A4CYP2D6GHSR
SCHEMBL1704865 0.82 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2GHSR
SCHEMBL4180898 0.80 MLNR (0.76) MLNRCYP3A4CYP2D6KCNH2GHSR
SCHEMBL1704458 0.78 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL3921210 0.76 KDM4E (0.39) MLNRCYP3A4
SCHEMBL3924366 0.76 KDM4E (0.39) MLNRCYP3A4
SCHEMBL3913756 0.74 GBA1 (0.41)
SCHEMBL1704619 0.73 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2GHSR
SCHEMBL1703969 0.72 MLNR (0.63) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4183557 0.71 MLNR (0.77) MLNRCYP3A4CYP2D6KCNH2GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907374-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-09 EP disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed