SCHEMBL4596941

SCHEMBL4596941

C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2Cl)CC[N+]1(C(=O)[O-])C(C)(C)C

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MLNR O43193 20/20 0.69
CYP3A4 P08684 7/20 0.56
CYP2D6 P10635 2/20 0.56
KCNH2 Q12809 1/20 0.56
CYP1A2 P05177 1/20 0.41
GHSR Q92847 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920664 0.82 MLNR (0.51) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1704149 0.82 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL3913651 0.81 MLNR (0.44) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL4188248 0.80 MLNR (0.75) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1705080 0.80 MLNR (0.70) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1705081 0.76 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL3912866 0.76 MLNR (0.42) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL3924957 0.74 EPHX2 (0.38) MLNR
SCHEMBL14618671 0.73 MLNR (0.84) MLNRCYP3A4CYP2D6KCNH2CYP1A2
Camicinal SCHEMBL1703910 0.72 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907374-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-09 EP disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed