SCHEMBL4597013

SCHEMBL4597013

CC1CN(Cc2ccc(C(C)(C)C(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CC(C)N1C(=O)O

nearest known ligand 0.79

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MLNR O43193 17/20 0.79
CYP3A4 P08684 7/20 0.79
CYP2D6 P10635 2/20 0.48
GHSR Q92847 1/20 0.48
FAAH O00519 1/20 0.44
PRKAB2 O43741 2/20 0.44
PRKAG1 P54619 2/20 0.44
PRKAA2 P54646 2/20 0.44
PRKAA1 Q13131 2/20 0.44
PRKAG3 Q9UGI9 2/20 0.44
PRKAG2 Q9UGJ0 2/20 0.44
PRKAB1 Q9Y478 2/20 0.44
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4175700 1.00 MLNR (0.79) MLNRCYP3A4CYP2D6GHSRFAAH
SCHEMBL1704816 0.90 MLNR (0.74) MLNRCYP3A4CYP2D6GHSRPRKAB2
SCHEMBL1704589 0.88 MLNR (1.00) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4180898 0.86 MLNR (0.76) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL4185918 0.85 MLNR (0.77) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4183557 0.84 MLNR (0.77) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL1704464 0.78 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL14618440 0.77 MLNR (0.80) MLNRCYP3A4CYP2D6GHSR
SCHEMBL1704684 0.77 MLNR (0.71) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4597664 0.77 MLNR (0.82) MLNRCYP3A4CYP2D6GHSRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101258143-B Benzylpiperazine derivatives and their medical use GLAXO GROUP LTD 2012-12-26 CN disclosed
EP-1907374-A2 COMPOUNDS GLAXO GROUP LIMITED (GB) 2008-04-09 EP disclosed
WO-2007012479-A2 BENZYLPIPERAZINE DERIVATES AND THEIR MEDICAL USE GLAXO GROUP LIMITED (GB) 2007-02-01 WO disclosed