SCHEMBL4601049

SCHEMBL4601049

CSC(=S)N(C)N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cystogon SCHEMBL220119 0.73
Cystogon SCHEMBL28739900 0.71
SCHEMBL8986738 0.69
SCHEMBL8986695 0.69
SCHEMBL28440085 0.69
SCHEMBL28857712 0.69
SCHEMBL27464692 0.69
SCHEMBL20923539 0.69
SCHEMBL14281225 0.67
SCHEMBL20561014 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307239-A4 RADIOPHARMACEUTICAL FOR DIAGNOSTIC IMAGING CONTAINING A TECHNETIUM-99M NITRIDE HETEROCOMPLEX NIHON MEDIPHYSICS CO LTD (JP) 2005-01-26 EP claimed
US-20040018147-A1 Radiopharmaceutical for diagnostic imaging containing a technetium-99m nitride heterocomplex NIHON MEDI-PHYSICS CO., LTD. (JP) 2004-01-29 US claimed
EP-0949265-B1 RADIOACTIVE TRANSITION METAL NITRIDE HETERO-COMPLEX NIHON MEDIPHYSICS CO LTD (JP) 2003-05-07 EP claimed
EP-1307239-A1 RADIOPHARMACEUTICAL FOR DIAGNOSTIC IMAGING CONTAINING A TECHNETIUM-99M NITRIDE HETEROCOMPLEX Nihon Medi-Physics Co., Ltd. (JP) 2003-05-07 EP claimed
US-20020048549-A1 Radioactive transition metal nitride heterocomplex DUATTI ADRIANO (IT) 2002-04-25 US claimed
WO-2002009771-A1 RADIOPHARMACEUTICAL FOR DIAGNOSTIC IMAGING CONTAINING A TECHNETIUM-99M NITRIDE HETEROCOMPLEX NIHON MEDI-PHYSICS CO., LTD. (JP) 2002-02-07 WO claimed
CN-1322727-A Tc-99m labelled Tc-N nucleated isonitrile compound and its preparation and application UNIV BEIJING NORMAL (CN) 2001-11-21 CN claimed
US-6270745-B1 FROM A BIS(PHOSPHINOALKYL) SULFIDE OR AMINE NIHON MEDI-PHYSICS CO., LTD. (JP) 2001-08-07 US claimed
EP-0596037-B1 RADIOPHARMACEUTICAL PRODUCT HAVING IN PARTICULAR A CEREBRAL TROPISM COMPRISING A TRANSITION METAL NITRIDE COMPLEX, AND PREPARATION METHOD THEREFOR CIS BIO INT (FR) 2001-05-02 EP claimed
EP-0949265-A1 RADIOACTIVE TRANSITION METAL NITRIDE HETERO-COMPLEX Nihon Medi-Physics Co., Ltd. (JP) 1999-10-13 EP claimed
EP-0596037-A1 RADIOPHARMACEUTICAL PRODUCT HAVING IN PARTICULAR A CEREBRAL TROPISM COMPRISING A TRANSITION METAL NITRIDE COMPLEX, AND PREPARATION METHOD THEREFOR CIS BIO INTERNATIONAL (FR) 1994-05-11 EP claimed
US-5288476-A Technetium or rhenium complexed with dithiocarbamate ligands CIS BIO INTERNATIONAL (FR) 1994-02-22 US claimed
EP-0445190-B1 PHARMACEUTICAL PRODUCT HAVING, IN PARTICULAR, A CARDIAC TROPISM COMPRISING A NITRURO COMPLEX OF A TRANSITION METAL AND PROCESS FOR PREPARATION THEREOF CIS BIO INTERNATIONAL (FR) 1993-09-15 EP claimed
WO-1993001839-A1 RADIOPHARMACEUTICAL PRODUCT HAVING IN PARTICULAR A CEREBRAL TROPISM COMPRISING A TRANSITION METAL NITRIDE COMPLEX, AND PREPARATION METHOD THEREFOR CIS BIO INTERNATIONAL (FR) 1993-02-04 WO claimed
WO-1990006137-A1 PHARMACEUTICAL PRODUCT HAVING, IN PARTICULAR, A CARDIAC TROPISM COMPRISING A NITRURO COMPLEX OF A TRANSITION METAL AND PROCESS FOR PREPARATION THEREOF CIS BIO INTERNATIONAL (FR) 1990-06-14 WO claimed
EP-3554559-B1 METHOD FOR LABELING OF SENSITIVE AND THERMOSENSITIVE TARGETING BIOMOLECULES WITH TECHNETIUM BASED COMPOUNDS BRACCO IMAGING SPA (IT) 2022-02-02 EP disclosed
CN-107840312-B Method for removing mercury in acid making process by lead-zinc smelting flue gas 云南兴贤环保科技有限公司 2020-05-08 CN disclosed
EP-0445190-B1 PHARMACEUTICAL PRODUCT HAVING, IN PARTICULAR, A CARDIAC TROPISM COMPRISING A NITRURO COMPLEX OF A TRANSITION METAL AND PROCESS FOR PREPARATION THEREOF CIS BIO INTERNATIONAL (FR) 1993-09-15 EP disclosed
WO-1993001839-A1 RADIOPHARMACEUTICAL PRODUCT HAVING IN PARTICULAR A CEREBRAL TROPISM COMPRISING A TRANSITION METAL NITRIDE COMPLEX, AND PREPARATION METHOD THEREFOR CIS BIO INTERNATIONAL (FR) 1993-02-04 WO disclosed
US-4064262-A S-methyl 3-furfurylidene-2-methyl-dithiocarbazate and its use as a fungicide ICI AUSTRALIA LIMITED (AU) 1977-12-20 US disclosed