SCHEMBL4601174

SCHEMBL4601174

COc1cc(NC(=O)c2ccnc3ccccc23)cc(OC)c1OC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.62
GAK O14976 1/20 0.60
RIPK2 O43353 1/20 0.60
COQ8A Q8NI60 1/20 0.60
NLK Q9UBE8 1/20 0.60
MAPT P10636 5/20 0.58
HSD17B10 Q99714 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
POLB P06746 3/20 0.56
HTT P42858 2/20 0.56
LMNA P02545 2/20 0.53
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
ATM Q13315 2/20 0.53
ABCB1 P08183 1/20 0.53
ABCG2 Q9UNQ0 1/20 0.53
ALDH1A1 P00352 2/20 0.53
PKM P14618 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
MEN1 O00255 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1336449 0.81 SMN1; SMN2 (0.57) SMN1; SMN2GAKRIPK2COQ8ANLK
SCHEMBL4601893 0.81 GRM4 (0.62) SMN1; SMN2MAPTPOLBALDH1A1TDP1
SCHEMBL10061503 0.80 MAPT (0.77) MAPTPOLBHTTLMNAATM
SCHEMBL379808 0.79 CYP3A4 (0.60) MAPTL3MBTL1HTTNPSR1ALDH1A1
SCHEMBL10061786 0.79 MAPT (0.65) SMN1; SMN2MAPTPOLBHTTLMNA
SCHEMBL28579647 0.77 KDM4E (0.59) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL29886180 0.77 KDM4E (0.59) SMN1; SMN2MAPTPOLBALDH1A1MEN1
SCHEMBL8130849 0.76 ABCB1 (0.58) MAPTMAPK1ABCB1ABCG2KMT2A
SCHEMBL20945452 0.75 SMN1; SMN2 (0.68) SMN1; SMN2MAPTPOLBHTTLMNA
SCHEMBL11459070 0.75 HTT (0.73) SMN1; SMN2MAPTHTTLMNAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912970-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL Bayer Schering Pharma Aktiengesellschaft (DE) 2008-04-23 EP disclosed
WO-2007017289-A2 ACYLTRYPTOPHANOLS FOR FERTILITY CONTROL BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-02-15 WO disclosed