SCHEMBL4606764

SCHEMBL4606764

O=C(S)C1=NN(c2ccc(Cl)cc2Cl)C(c2ccc(F)cc2)C1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.57
CNR2 P34972 5/20 0.57
NR3C2 P08235 5/20 0.48
EGFR P00533 1/20 0.40
MARS1 P56192 1/20 0.39
PGR P06401 1/20 0.39
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605995 0.93 CNR1 (0.64) CNR1CNR2NR3C2EGFR
SCHEMBL2021047 0.90 CNR1 (0.58) CNR1CNR2NR3C2EGFRMARS1
SCHEMBL2017880 0.90 CNR1 (0.58) CNR1CNR2NR3C2EGFRMARS1
SCHEMBL14621870 0.90 CNR1 (0.58) CNR1CNR2NR3C2EGFRMARS1
SCHEMBL4607833 0.90 CNR1 (0.58) CNR1CNR2NR3C2EGFR
SCHEMBL14396247 0.89 CNR1 (0.57) CNR1CNR2NR3C2EGFRMARS1
Hydrochloric Acid SCHEMBL2021048 0.89 CNR1 (0.57) CNR1CNR2NR3C2EGFRMARS1
SCHEMBL4607251 0.89 CNR1 (0.57) CNR1CNR2NR3C2EGFR
SCHEMBL4607305 0.86 CNR1 (0.54) CNR1CNR2EGFRMAOB
SCHEMBL2021086 0.86 CNR1 (0.56) CNR1CNR2NR3C2EGFRMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1946777-A1 Substituted pyrazoline for preventing weight gain Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP claimed
EP-1946778-A1 Active substance combination for the treatment of diabetes Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP claimed
EP-1743887-A1 Thiocarbonyl-substituted pyrazoline compounds, their preparation and use as CB1 modulators LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-01-17 EP claimed
EP-1946777-A1 Substituted pyrazoline for preventing weight gain Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed
EP-1946778-A1 Active substance combination for the treatment of diabetes Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed
EP-1743887-A1 Thiocarbonyl-substituted pyrazoline compounds, their preparation and use as CB1 modulators LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-01-17 EP disclosed