SCHEMBL4606989

SCHEMBL4606989

Nc1c(Br)cc(C[C@@H](NC(=O)N2CCC(n3c(=O)[nH]c4c5ccccc5ncc43)CC2)C(=O)N2CCC(N3CCCCC3)CC2)cc1Br

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 17/20 0.64
CYP3A4 P08684 10/20 0.64
RAMP1 O60894 1/20 0.52
CALCA P06881 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144584 0.91 CALCRL (0.53) CALCRLCYP3A4RAMP1CALCA
SCHEMBL2026964 0.91 CALCRL (0.53) CALCRLCYP3A4RAMP1CALCA
SCHEMBL3903201 0.85 CALCRL (0.60) CALCRLCYP3A4RAMP1CALCA
SCHEMBL2031664 0.84 CALCRL (0.46) CALCRLCYP3A4RAMP1CALCA
SCHEMBL3900985 0.84 CALCRL (0.47) CALCRLCYP3A4RAMP1CALCA
SCHEMBL3277961 0.82 CALCRL (0.53) CALCRLCYP3A4
SCHEMBL3279641 0.81 CALCRL (0.53) CALCRLCYP3A4CALCA
SCHEMBL4150835 0.81 CALCRL (0.75) CALCRLCYP3A4RAMP1
SCHEMBL13313769 0.81 CALCRL (0.53) CALCRLCYP3A4RAMP1CALCA
SCHEMBL13313782 0.81 CALCRL (0.46) CALCRLCYP3A4RAMP1CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP claimed
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP disclosed