SCHEMBL4607152

SCHEMBL4607152

O=C(O)C1=NN(c2ccc(Cl)cc2Cl)C(c2cc(CCl)cs2)C1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.44
CNR2 P34972 5/20 0.44
PTGS2 P35354 2/20 0.37
PDE5A O76074 1/20 0.37
GRM5 P41594 8/20 0.36
NOTUM Q6P988 1/20 0.35
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4604892 0.86 CNR1 (0.46) CNR1CNR2PTGS2PDE5AGRM5
SCHEMBL4606961 0.84 CNR1 (0.57) CNR1CNR2
SCHEMBL4604890 0.81 CNR1 (0.47) CNR1CNR2PTGS2PDE5ANOTUM
SCHEMBL4606276 0.79 CNR1 (0.46) CNR1CNR2PTGS2PDE5ANOTUM
SCHEMBL1748630 0.79 CNR1 (0.65) CNR1CNR2PDE5ANOTUM
SCHEMBL1748594 0.79 CNR1 (0.65) CNR1CNR2PDE5ANOTUM
SCHEMBL1748655 0.79 CNR1 (0.65) CNR1CNR2PDE5ANOTUM
SCHEMBL31589469 0.79 CNR1 (0.65) CNR1CNR2PDE5ANOTUM
Hydrochloric Acid SCHEMBL1749138 0.78 CNR1 (0.64) CNR1CNR2PTGS2PDE5ANOTUM
SCHEMBL2021231 0.76 CNR1 (0.59) CNR1CNR2PDE5ANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1946777-A1 Substituted pyrazoline for preventing weight gain Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed
EP-1946778-A1 Active substance combination for the treatment of diabetes Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed