SCHEMBL4607240

SCHEMBL4607240

CC(C)S(=O)(=O)N[C@@H]1CCC[C@H]1c1ccc(-c2ccc(C#N)cc2)cc1

nearest known ligand 0.93

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 14/20 0.93
GRIA2 P42262 8/20 0.69
KCNH2 Q12809 4/20 0.69
GRIA1 P42261 2/20 0.46
GRIA3 P42263 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608569 1.00 GRIA4 (0.93) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL4609445 0.96 GRIA4 (1.00) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL4608206 0.96 GRIA4 (1.00) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL2212874 0.86 GRIA2 (0.74) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL2212870 0.86 GRIA2 (0.74) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL13140825 0.86 GRIA2 (0.74) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL3186437 0.85 GRIA4 (0.67) GRIA4GRIA2KCNH2GRIA1GRIA3
SCHEMBL14141257 0.85 GRIA4 (0.67) GRIA4GRIA2KCNH2
SCHEMBL4607516 0.85 GRIA4 (0.67) GRIA4GRIA2KCNH2
SCHEMBL4608046 0.85 GRIA4 (0.84) GRIA4GRIA2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246797-B1 CYCLOPENTYL SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2008-07-23 EP claimed