SCHEMBL4608743

SCHEMBL4608743

CCCNC(=O)N(c1ccc(C)cc1)c1ccnc(NC(C)COC)n1

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 18/20 0.61
HCAR3 P49019 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608745 1.00 MAPK14 (0.61) MAPK14HCAR3
SCHEMBL4610274 0.94 MAPK14 (0.60) MAPK14
SCHEMBL4610270 0.94 MAPK14 (0.60) MAPK14
SCHEMBL4608723 0.92 MAPK14 (0.64) MAPK14HCAR3
SCHEMBL4608725 0.92 MAPK14 (0.64) MAPK14HCAR3
SCHEMBL4608407 0.91 MAPK14 (0.70) MAPK14
SCHEMBL4609124 0.91 MAPK14 (0.58) MAPK14
SCHEMBL4609120 0.91 MAPK14 (0.58) MAPK14
SCHEMBL4608404 0.91 MAPK14 (0.70) MAPK14
SCHEMBL4624341 0.91 MAPK14 (0.57) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449474-B2 Tri-substituted ureas as cytokine inhibitors THE PROCTER & GAMBLE COMPANY (US) 2008-11-11 US claimed
EP-1747204-B1 TRI-SUBSTITUTED UREAS AS CYTOKINE INHIBITORS PROCTER & GAMBLE (US) 2008-07-30 EP claimed
EP-1747204-A1 TRI-SUBSTITUTED UREAS AS CYTOKINE INHIBITORS The Procter and Gamble Company (US) 2007-01-31 EP claimed
WO-2005105758-A1 TRI-SUBSTITUTED UREAS AS CYTOKINE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2005-11-10 WO claimed