Triaziquone

Triaziquone

SCHEMBL4608905

O=C(O)O.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.43
MAPT P10636 4/20 0.41
HTT P42858 2/20 0.41
TP53 P04637 1/20 0.41
STAT3 P40763 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NSD2 O96028 4/20 0.36
APAF1 O14727 3/20 0.36
HKDC1 Q2TB90 3/20 0.36
TDP2 O95551 2/20 0.36
KMT2A Q03164 3/20 0.34
GALK1 P51570 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
BLM P54132 1/20 0.34
ATM Q13315 1/20 0.34
NOD2 Q9HC29 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL8926769 0.94 DNMT1 (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL9678206 0.93 DNMT1 (0.39) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL16419 0.92 MAPT (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL11422311 0.92 MAPT (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL4334317 0.91 DNMT1 (0.40) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL738610 0.90 DNMT1 (0.42) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL3101456 0.90 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL6000230 0.90 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL5054475 0.90 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3
Triaziquone SCHEMBL7088197 0.90 DNMT1 (0.47) DNMT1MAPTHTTTP53STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070031910-A1 Method of stabilizing sample ARKRAY, INC. (JP) 2007-02-08 US claimed
EP-1628134-A1 METHOD OF STABILIZING SAMPLE ARKRAY, Inc. (JP) 2006-02-22 EP claimed
WO-2024036507-A1 ELECTROCHEMICAL DEVICE AND ELECTRONIC DEVICE 宁德新能源科技有限公司 2024-02-22 WO disclosed
CN-112300435-A Environment-friendly polyurethane foaming agent and preparation method thereof 宋庆红 2021-02-02 CN disclosed
EP-1443327-B1 Biochemical and immunochemical assay device DIAMATRIX LTD (GB) 2008-07-30 EP disclosed
US-7303923-B2 Biochemical and immunochemical assay device DIAMATRIX LIMITED (GB) 2007-12-04 US disclosed
US-20070031910-A1 Method of stabilizing sample ARKRAY, INC. (JP) 2007-02-08 US disclosed
CN-1795381-A Method for stabilizing hemolyzed sample ARKRAY INC (JP) 2006-06-28 CN disclosed
EP-1628134-A1 METHOD OF STABILIZING SAMPLE ARKRAY, Inc. (JP) 2006-02-22 EP disclosed
EP-1443327-A2 Biochemical and immunochemical assay device DIAMATRIX LIMITED (GB) 2004-08-04 EP disclosed
EP-0968426-B1 BIOCHEMICAL AND IMMUNOCHEMICAL ASSAY DEVICE DIAMATRIX LTD (GB) 2004-04-07 EP disclosed
US-4794077-A DIAGNOSIS BIOSCIENCES CORPORATION OF TEXAS (US) 1988-12-27 US disclosed
EP-0284429-A2 Antibodies to human cancer nucleolar antigen pl20, corresponding cell lines, and their preparation and use in the detection of human cancer cells BIOSCIENCES CORPORATION OF TEXAS (US) 1988-09-28 EP disclosed
EP-0259949-A2 Method of improving optical clarity in reconstituted lyophilized products TECHNICON INSTRUMENTS CORPORATION(a Delaware corporation) (US) 1988-03-16 EP disclosed
EP-0226468-A2 Detection of human cancer cells with antibodies to human cancer nucleolar antigen p145 ONCOS, LTD. (US) 1987-06-24 EP disclosed
EP-0016573-B1 ENZYME REFERENCE COMPOSITION BECKMAN INSTRUMENTS, INC. (US) 1984-06-13 EP disclosed
US-4448890-A DIAGNOSTIC KITS BAYLOR COLLEGE OF MEDICINE (US) 1984-05-15 US disclosed
US-4325832-A POLYOXYALKYLENE GLYCOL, PROTEIN BECKMAN INSTRUMENTS, INC. (US) 1982-04-20 US disclosed
EP-0016573-A1 Enzyme reference composition BECKMAN INSTRUMENTS, INC. (US) 1980-10-01 EP disclosed
US-4089747-A OXIDATION OF DYE-PROVIDING MATERIALS, A SULFONYL HYDRAZONE AND A COUPLER OR A TRIARYLIMIDAZOLE EASTMAN KODAK COMPANY (US) 1978-05-16 US disclosed