SCHEMBL4612416

SCHEMBL4612416

CN1C(=O)C(c2c[c]ccc2)(C2CCCCC2)N=C1N

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.76
BACE2 Q9Y5Z0 14/20 0.76
APP P05067 3/20 0.76
CTSD P07339 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189524 0.86 BACE1 (1.00) BACE1BACE2APPCTSD
SCHEMBL8231970 0.85 BACE1 (0.97) BACE1BACE2APPCTSD
SCHEMBL4599277 0.79 BACE1 (0.72) BACE1BACE2APPCTSD
SCHEMBL4599272 0.79 BACE1 (0.72) BACE1BACE2APPCTSD
Trifluoroacetic Acid SCHEMBL4229079 0.77 BACE1 (0.80) BACE1BACE2APPCTSD
SCHEMBL4611233 0.76 BACE1 (0.71) BACE1BACE2APPCTSD
SCHEMBL5146663 0.74 BACE1 (0.77) BACE1BACE2APPCTSD
SCHEMBL5522143 0.74 BACE1 (0.73) BACE1BACE2APPCTSD
SCHEMBL8414534 0.73 BACE1 (0.63) BACE1BACE2APPCTSD
SCHEMBL4708358 0.73 BACE1 (0.74) BACE1BACE2APPCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910309-A2 CYCLOALKYL AMINO-HYDANTOIN COMPOUNDS AND USE THEREOF FOR ß-SECRETASE MODULATION Wyeth (US) 2008-04-16 EP claimed
WO-2007016012-A2 CYCLOALKYL AMINO-HYDANTOIN COMPOUNDS AND USE THEREOF FOR β-SECRETASE MODULATION WYETH (US) 2007-02-08 WO claimed