SCHEMBL4618979

SCHEMBL4618979

OCc1cc([C@H]2O[C@@H](n3cnc4c(N[C@H](CO)Cc5ccccc5)nc(Cl)nc43)[C@H](O)[C@@H]2O)on1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.72
ADORA3 P0DMS8 5/20 0.49
ADORA2A P29274 4/20 0.49
HTR2C P28335 1/20 0.49
ADORA2B P29275 1/20 0.48
NT5E P21589 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2809155 0.94 ADORA1 (0.70) ADORA1ADORA3ADORA2AHTR2CADORA2B
SCHEMBL2832621 0.94 ADORA1 (0.70) ADORA1ADORA3ADORA2AHTR2CADORA2B
SCHEMBL3913337 0.94 ADORA1 (0.70) ADORA1ADORA3ADORA2AHTR2CADORA2B
SCHEMBL4230273 0.94 ADORA1 (0.70) ADORA1ADORA3ADORA2AHTR2CADORA2B
SCHEMBL2805070 0.84 ADORA2A (0.54) ADORA1ADORA3ADORA2AADORA2BNT5E
Trifluoroacetic Acid SCHEMBL6839083 0.84 ADORA1 (0.51) ADORA1ADORA3ADORA2AHTR2CADORA2B
SCHEMBL6838893 0.84 ADORA1 (0.58) ADORA1ADORA3ADORA2AADORA2BNT5E
SCHEMBL6841625 0.84 ADORA2A (0.56) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL6876893 0.84 ADORA1 (0.56) ADORA1ADORA3ADORA2AADORA2BNT5E
SCHEMBL6573910 0.82 ADORA1 (0.57) ADORA1ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044070-B1 PURINE DERIVATIVES AS A2A AGONISTS NOVARTIS AG (CH) 2012-08-22 EP disclosed
EP-1889846-A1 Purine derivatives as A2a agonists Novartis AG (CH) 2008-02-20 EP disclosed