SCHEMBL4619623

SCHEMBL4619623

CC(C)COC(=O)NCc1nc(CN(CC(F)(F)F)c2ccc(C#N)c(C(F)(F)F)c2)no1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AR P10275 12/20 0.44
PGR P06401 1/20 0.44
FPR2 P25090 1/20 0.33
SCN9A Q15858 1/20 0.33
S1PR1 P21453 1/20 0.32
XDH P47989 2/20 0.31
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13777361 0.88 AR (0.42) ARPGR
SCHEMBL4153666 0.87 AR (0.45) ARPGR
SCHEMBL4153588 0.85 AR (0.43) ARPGRFPR2SCN9A
SCHEMBL13777376 0.82 AR (0.41) ARPGRFPR2SCN9A
SCHEMBL4145273 0.82 AR (0.39) ARPGRFPR2SCN9A
SCHEMBL4147163 0.81 AR (0.41) ARPGRS1PR1
SCHEMBL4145386 0.80 AR (0.44) ARPGR
SCHEMBL13777375 0.80 AR (0.41) ARPGR
SCHEMBL4146432 0.79 AR (0.46) ARPGR
SCHEMBL4158830 0.79 AR (0.42) ARPGRFPR2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888512-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-20 EP disclosed
WO-2006133216-A2 4-SUBSTITUTED ARYLAMINE DERIVATIVES AND THEIR USE IN PHARMACEUTICAL COMPOSITIONS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed