SCHEMBL462123

SCHEMBL462123

CCCCCNC(=S)NCCCCC

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.55
EPHX1 P07099 6/20 0.54
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CASP2 P42575 1/20 0.48
ALDH1A1 P00352 2/20 0.48
TSHR P16473 1/20 0.48
CYP3A4 P08684 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11594937 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11596495 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL8979287 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL1273832 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11593203 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11596219 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL5081267 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11594414 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11595110 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A
SCHEMBL11596178 0.97 EPHX1 (0.58) EPHX2EPHX1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 147 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024006252-A1 DUAL INHIBITION OF MDM2 AND EIF2-ALPHA INDUCES CELL DEATH IN MULTIPLE CANCER CELL TYPES THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2024-01-04 WO claimed
US-7385008-B2 Abrasion resistant elastomeric compositions EXXONMOBILE CHEMICAL PATENTS INC. (US) 2008-06-10 US claimed
US-20080033101-A1 Abrasion Resistant Elastomeric Compositions EXXONMOBIL CHEMICAL PATENTS INC. 2008-02-07 US claimed
US-7300981-B2 Abrasion resistant elastomeric compositions EXXONMOBIL CHEMICAL PATENTS INC. (US) 2007-11-27 US claimed
EP-1501874-A4 ABRASION RESISTANT ELASTOMERIC COMPOSITIONS EXXONMOBIL CHEM PATENTS INC (US) 2005-08-31 EP claimed
CN-1642988-A Abrasion resistant elastomeric compositions EXXONMOBIL CHEM PATENTS INC (US) 2005-07-20 CN claimed
JP-2005520022-A 2005-07-07 JP claimed
US-20050085594-A1 Abrasion resistant elastomeric compositions EXXONMOBIL CHEMICAL PATENTS INC. 2005-04-21 US claimed
EP-1501874-A1 ABRASION RESISTANT ELASTOMERIC COMPOSITIONS Exxonmobil Chemical Patents Inc. (US) 2005-02-02 EP claimed
WO-2003078475-A1 ABRASION RESISTANT ELASTOMERIC COMPOSITIONS EXXONMOBIL CHEMICAL PATENTS, INC. (US) 2003-09-25 WO claimed
EP-0643646-B1 THERMOSENSITIVE RECORDING ELEMENT INT PAPER CO (US) 1997-03-12 EP claimed
US-5610118-A LAYERS WITH ELECTRON DONATING DYE PRECURSOR AND ELECTRON ACCEPTING COMPOUND; THERMAL PRINTING INTERNATIONAL PAPER COMPANY (US) 1997-03-11 US claimed
EP-0609323-B1 THERMOSENSITIVE RECORDING ELEMENT HAVING IMPROVED SMOOTHNESS CHARACTERISTICS INT PAPER CO (US) 1996-06-19 EP claimed
US-5380694-A Thermosensitive recording element INTERNATIONAL PAPER COMPANY (US) 1995-01-10 US claimed
US-5250717-A Reacting thiourea with unsubstituted or mono-, di- or tri-alkyl substituted m-phenylenediamines with controlled heating ETHYL CORPORATION (US) 1993-10-05 US claimed
WO-1993008031-A1 ABRASION RESISTANT, THERMOSENSITIVE RECORDING ELEMENT INTERNATIONAL PAPER COMPANY (US) 1993-04-29 WO claimed
EP-0538639-A1 Thermosensitive recording element E.I. DU PONT DE NEMOURS & COMPANY INCORPORATED (US) 1993-04-28 EP claimed
JP-1123785-A None JP disclosed
US-4688058-A Thermal recording materials MITSUBISHI PAPER MILLS, LTD. (JP) 1987-08-18 US disclosed
US-4252963-A CYCLIZATION OF PHENYLTHIOUREAS WITH THIONYL CHLORIDE HOECHST AKTIENGESELLSCHAFT (DE) 1981-02-24 US disclosed