SCHEMBL4621743

SCHEMBL4621743

COc1nc(NCCO)nc(OC)c1NC(=O)c1csc(Oc2cc(Cl)ccc2C)n1.COc1nc(OCCO)nc(OC)c1NC(=O)c1csc(Oc2cc(C(C)(C)C)ccc2C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 5/20 0.37
POLB P06746 1/20 0.35
S1PR2 O95136 1/20 0.32
S1PR4 O95977 1/20 0.32
MDM2 Q00987 2/20 0.32
NR1I2 O75469 1/20 0.31
SYK P43405 1/20 0.31
IRAK1 P51617 1/20 0.31
CCR9 P51686 1/20 0.31
SCN9A Q15858 1/20 0.31
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
GNRHR P30968 2/20 0.30
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30
HPGD P15428 1/20 0.30
CACNA1F O60840 1/20 0.30
CHRM4 P08173 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4226409 0.91 IRAK4 (0.35) IRAK4POLBSYKGNRHRHPGD
SCHEMBL4229030 0.91 EDNRA (0.33) POLBNR1I2EDNRBEDNRA
SCHEMBL4232018 0.88 IRAK4 (0.43) IRAK4POLBMDM2SYKIRAK1
SCHEMBL4621267 0.86 GRM4 (0.36) NR1I2EDNRBEDNRA
SCHEMBL13743435 0.85 GNRHR (0.35) POLBNR1I2GNRHRHPGDCACNA1F
SCHEMBL4231634 0.84 GNRHR (0.42) POLBGAAGNRHRHPGDCACNA1F
SCHEMBL4236457 0.84 SYK (0.36) IRAK4POLBSYKIRAK1GNRHR
SCHEMBL4231659 0.83 NR1I2 (0.33) POLBNR1I2
SCHEMBL4233491 0.83 GRM4 (0.38) POLBNR1I2
SCHEMBL4233369 0.83 GNRHR (0.36) GAAGNRHRHPGDCACNA1FCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896465-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS Takeda Cambridge Limited (GB) 2008-03-12 EP claimed
WO-2007000582-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS TAKEDA CAMBRIDGE LIMITED (GB) 2007-01-04 WO claimed