SCHEMBL4624067

SCHEMBL4624067

Cc1cccc(Cl)c1C(=O)NC(Cc1ccc2nc(-c3c(C)cccc3C)ccc2c1)C(=O)O

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.80
ITGAV P06756 1/20 0.80
ITGA4 P13612 18/20 0.59
ITGB7 P26010 11/20 0.59
ITGA2 P17301 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3315868 0.97 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3314968 0.96 ITGB1 (0.87) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3314741 0.95 ITGB1 (0.76) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3318272 0.93 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3320790 0.93 ITGB1 (0.75) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3313255 0.92 ITGB1 (0.77) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL6139776 0.92 ITGB1 (0.77) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL8352229 0.89 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3313373 0.89 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3316398 0.89 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed
EP-1870402-A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors UCB Pharma, S.A. (BE) 2007-12-26 EP disclosed