SCHEMBL4625192

SCHEMBL4625192

Cn1nc(C(F)(F)F)c(-c2ccc3cc(CC(NC(=O)c4c(Cl)cccc4Cl)C(=O)O)ccc3n2)c1Cl

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.73
ITGAV P06756 1/20 0.73
ITGA4 P13612 19/20 0.51
ITGB7 P26010 18/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314948 0.95 ITGB1 (0.67) ITGB1ITGAVITGA4ITGB7
SCHEMBL4625313 0.87 ITGB1 (0.55) ITGB1ITGAVITGA4ITGB7
SCHEMBL3316398 0.85 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7
SCHEMBL8352229 0.85 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313373 0.85 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313356 0.85 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7
SCHEMBL3314805 0.84 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7
SCHEMBL3316590 0.82 ITGB1 (0.89) ITGB1ITGAVITGA4ITGB7
SCHEMBL3316443 0.82 ITGB1 (0.89) ITGB1ITGAVITGA4ITGB7
SCHEMBL3315868 0.82 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed
EP-1870402-A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors UCB Pharma, S.A. (BE) 2007-12-26 EP disclosed