SCHEMBL4626488

SCHEMBL4626488

COc1ccccc1Oc1ccc2cc(CC(NC(=O)c3c(Cl)cccc3Cl)C(=O)O)ccc2n1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.64
ITGAV P06756 4/20 0.64
ITGA4 P13612 15/20 0.53
ITGB7 P26010 9/20 0.53
ITGA5 P08648 4/20 0.50
ITGB3 P05106 3/20 0.50
ITGA2 P17301 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4624998 0.93 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL4624246 0.93 ITGB1 (0.64) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL5173381 0.90 ITGB1 (0.72) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3317334 0.88 ITGB1 (0.69) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL4625183 0.87 ITGB1 (0.71) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL4627182 0.86 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3318793 0.86 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3314866 0.86 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3313117 0.86 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL4625259 0.85 ITGB1 (0.67) ITGB1ITGAVITGA4ITGB7ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed
EP-1870402-A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors UCB Pharma, S.A. (BE) 2007-12-26 EP disclosed