Predicted protein targets (top 17)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | P2RX4 | Q99571 | 4/20 | 0.41 |
| ▸ | NOTUM | Q6P988 | 1/20 | 0.40 |
| ▸ | ALOX12 | P18054 | 1/20 | 0.40 |
| ▸ | HSD17B3 | P37058 | 1/20 | 0.38 |
| ▸ | TSHR | P16473 | 2/20 | 0.37 |
| ▸ | HTT | P42858 | 2/20 | 0.36 |
| ▸ | ALDH1A1 | P00352 | 1/20 | 0.36 |
| ▸ | GAA | P10253 | 1/20 | 0.36 |
| ▸ | ADAMTS4 | O75173 | 1/20 | 0.36 |
| ▸ | MAPT | P10636 | 2/20 | 0.36 |
| ▸ | TP53 | P04637 | 1/20 | 0.36 |
| ▸ | POLB | P06746 | 1/20 | 0.36 |
| ▸ | SMN1; SMN2 | Q16637 | 2/20 | 0.36 |
| ▸ | SLC22A12 | Q96S37 | 1/20 | 0.35 |
| ▸ | LMNA | P02545 | 1/20 | 0.35 |
| ▸ | NPSR1 | Q6W5P4 | 1/20 | 0.35 |
| ▸ | THRB | P10828 | 1/20 | 0.34 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL4626535 | 1.00 | P2RX4 (0.41) | P2RX4NOTUMALOX12HSD17B3TSHR | |
| SCHEMBL16095343 | 0.71 | NOTUM (0.40) | NOTUMHSD17B3ALDH1A1MAPT | |
| SCHEMBL16095342 | 0.71 | NOTUM (0.40) | NOTUMHSD17B3ALDH1A1MAPT | |
| SCHEMBL8177425 | 0.69 | ABCG2 (0.37) | P2RX4NOTUMHSD17B3TSHRHTT | |
| SCHEMBL4444354 | 0.67 | NOTUM (0.53) | P2RX4NOTUMHSD17B3TSHRHTT | |
| Acetic Acid SCHEMBL27604418 | 0.67 | NOTUM (0.49) | P2RX4NOTUMHSD17B3HTTALDH1A1 | |
| Hydrochloric Acid SCHEMBL23320556 | 0.66 | NOTUM (0.51) | P2RX4NOTUMHSD17B3TSHRHTT | |
| Acetic Acid SCHEMBL5469518 | 0.66 | NOTUM (0.47) | P2RX4NOTUMHSD17B3HTTALDH1A1 | |
| SCHEMBL12660327 | 0.65 | ABCG2 (0.39) | P2RX4NOTUMALOX12HSD17B3TSHR | |
| SCHEMBL17603549 | 0.65 | NOTUM (0.49) | NOTUMLMNANPSR1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-1592801-A4 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | ADVANCED PROTEOME THERAPEUTICS (US) | 2008-04-30 | — | — | EP | claimed |
| EP-1592801-A2 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | Advanced Proteome Therapeutics Inc. (US) | 2005-11-09 | — | — | EP | claimed |
| WO-2004066917-A2 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | ADVANCED PROTEOME THERAPEUTICS, INC (US) | 2004-08-12 | — | — | WO | claimed |
| EP-1592801-A4 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | ADVANCED PROTEOME THERAPEUTICS (US) | 2008-04-30 | — | — | EP | disclosed |
| EP-1592801-A2 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | Advanced Proteome Therapeutics Inc. (US) | 2005-11-09 | — | — | EP | disclosed |
| WO-2004066917-A2 | TANDEM ANALYSES OF NONCOVALENTLY DRIVEN EFFECTORS FOR MODULATORY MAPPING OF ACTIVITIES OF PROTEIN SITES | ADVANCED PROTEOME THERAPEUTICS, INC (US) | 2004-08-12 | — | — | WO | disclosed |