SCHEMBL462859

SCHEMBL462859

N#Cc1cc(F)cc([C@H]2CC(F)(F)CN2c2ccn3nccc3n2)c1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.54
JAK2 O60674 2/20 0.43
ROS1 P08922 2/20 0.38
GRM5 P41594 1/20 0.33
FADS1 O60427 1/20 0.31
IDH1 O75874 1/20 0.31
RIPK1 Q13546 1/20 0.31
USP30 Q70CQ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460709 0.84 NTRK1 (0.57) NTRK1JAK2ROS1
SCHEMBL460710 0.84 NTRK1 (0.57) NTRK1JAK2ROS1
SCHEMBL462737 0.79 NTRK1 (0.59) NTRK1JAK2
SCHEMBL462170 0.75 NTRK1 (0.55) NTRK1JAK2
SCHEMBL460633 0.75 NTRK1 (0.55) NTRK1JAK2
SCHEMBL12477947 0.72 NTRK1 (0.45) NTRK1JAK2ROS1RIPK1
SCHEMBL12477980 0.71 NTRK1 (0.44) NTRK1JAK2RIPK1
SCHEMBL12477982 0.71 NTRK1 (0.44) NTRK1JAK2RIPK1
SCHEMBL18863642 0.70 NTRK1 (1.00) NTRK1JAK2
SCHEMBL18863641 0.70 NTRK1 (1.00) NTRK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012034095-A1 COMPOUNDS AND COMPOSITIONS AS TRK INHIBITORS IRM LLC (BM) 2012-03-15 WO claimed