SCHEMBL4629115

SCHEMBL4629115

Cc1c(C)c(C)c(CC2=NCCN2)c(C)c1C.Cc1cc(C)c(C)c(CC2=NCCN2)c1C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.66
HTR1B P28222 9/20 0.66
TAAR1 Q96RJ0 6/20 0.61
ADRA2A P08913 6/20 0.60
ADRA2B P18089 5/20 0.60
ADRA2C P18825 5/20 0.60
ADRA1D P25100 5/20 0.60
ADRA1A P35348 5/20 0.60
ADRA1B P35368 5/20 0.60
HTR1A P08908 4/20 0.60
LMNA P02545 4/20 0.60
CYP2D6 P10635 4/20 0.60
TSHR P16473 4/20 0.60
CHRM2 P08172 2/20 0.60
CHRM1 P11229 2/20 0.60
HTR2A P28223 2/20 0.60
HTR2C P28335 2/20 0.60
DRD3 P35462 2/20 0.60
HTR2B P41595 2/20 0.60
TP53 P04637 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953962 0.97 HTR1D (0.70) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL684149 0.90 HTR1D (0.71) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL953214 0.89 HTR1D (0.62) HTR1DHTR1BTAAR1ADRA2AADRA2B
Oxymetazoline SCHEMBL4629825 0.83 HTR1D (0.86) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL953076 0.79 HTR1D (1.00) HTR1DHTR1BTAAR1ADRA2AADRA2B
Oxymetazoline SCHEMBL4630526 0.79 HTR1D (0.91) HTR1DHTR1BTAAR1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL7969470 0.78 HTR1D (0.97) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL22953216 0.77 HTR1D (0.78) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL953638 0.77 HTR1D (0.76) HTR1DHTR1BTAAR1ADRA2AADRA2B
SCHEMBL7982884 0.77 HTR1D (1.00) HTR1DHTR1BTAAR1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed