SCHEMBL4629641

SCHEMBL4629641

CCc1cccc(CC)c1Cc1ncc[nH]1.FC(F)(F)c1cccc(CC2=NCCN2)c1Cl

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 12/20 0.55
HTR1A P08908 2/20 0.55
NISCH Q9Y2I1 2/20 0.38
MAPK1 P28482 2/20 0.38
ADRA1A P35348 2/20 0.38
LMNA P02545 1/20 0.38
ADRA2A P08913 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
OPRM1 P35372 1/20 0.38
HTR1D P28221 1/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
P2RX7 Q99572 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953083 0.82 TAAR1 (0.68) TAAR1HTR1ANISCHMAPK1ADRA1A
SCHEMBL952681 0.74 TAAR1 (1.00) TAAR1HTR1AADRA2ACYP2D6ADRA2B
SCHEMBL953493 0.73 TAAR1 (1.00) TAAR1HTR1ANISCHMAPK1ADRA1A
SCHEMBL4629815 0.72 TAAR1 (0.46) TAAR1HTR1ANISCHADRA1AADRA2A
SCHEMBL26078566 0.71 TAAR1 (0.68) TAAR1HTR1ANISCHMAPK1ADRA1A
SCHEMBL955372 0.71 TAAR1 (0.80) TAAR1HTR1AADRA1AADRA2AADRA2B
SCHEMBL954867 0.70 TAAR1 (0.70) TAAR1HTR1ANISCHMAPK1ADRA1A
Naphazoline SCHEMBL9789833 0.70 TAAR1 (0.70) TAAR1HTR1ANISCHMAPK1ADRA1A
SCHEMBL4630336 0.70 TAAR1 (0.47) TAAR1HTR1ANISCHMAPK1ADRA1A
SCHEMBL953494 0.69 TAAR1 (1.00) TAAR1HTR1ANISCHMAPK1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981497-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085557-A2 USE OF SUBSTITUTED 2-IMIDAZOLE OF IMIDAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed