SCHEMBL4631779

SCHEMBL4631779

O=C1COC(CCN2CCC(O)(c3ccccc3)CC2)(c2ccc(Cl)c(Cl)c2)CN1Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.63
TACR2 P21452 3/20 0.48
TACR3 P29371 2/20 0.48
CCR5 P51681 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7749138 0.98 TACR1 (0.61) TACR1TACR2TACR3CCR5
SCHEMBL4630849 0.95 TACR1 (0.69) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750416 0.93 TACR1 (0.67) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7750422 0.93 TACR1 (0.67) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7772688 0.89 TACR1 (0.49) TACR1TACR2TACR3CCR5
SCHEMBL4629935 0.84 TACR1 (0.42) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7772689 0.83 TACR1 (0.45) TACR1TACR2TACR3CCR5
SCHEMBL4631333 0.83 TACR1 (0.66) TACR1TACR2TACR3CCR5
SCHEMBL4630133 0.82 TACR1 (0.55) TACR1TACR2TACR3CCR5
Hydrochloric Acid SCHEMBL7749196 0.82 TACR1 (0.65) TACR1TACR2TACR3CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1923391-A1 Substituted heterocyclic compounds, method for preparing same and pharmaceutical compositions containing them. sanofi-aventis (FR) 2008-05-21 EP disclosed
EP-1688416-A1 Substituted heterocyclic compounds, their process of preparation and pharmaceutical compositions containing them Sanofi-Aventis (FR) 2006-08-09 EP disclosed
EP-1340754-A1 Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them SANOFI-SYNTHELABO (FR) 2003-09-03 EP disclosed
EP-1156049-A1 Substituted heterocyclic compounds, their process of preparation and pharmaceutical compositions containing them SANOFI-SYNTHELABO (FR) 2001-11-21 EP disclosed
WO-1996023787-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI (FR) 1996-08-08 WO disclosed