SCHEMBL4632572

SCHEMBL4632572

COC(=O)c1sc(-n2cnc3ccc(OC[C@@]4(C(C)(C)C)CN(C(=O)O)CCO4)cc32)cc1O[C@H](C)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 16/20 0.58
PLK3 Q9H4B4 15/20 0.58
NEK2 P51955 3/20 0.53
PIK3CD O00329 2/20 0.53
NUAK1 O60285 2/20 0.53
PDGFRB P09619 2/20 0.53
PIM1 P11309 2/20 0.53
KDR P35968 2/20 0.53
CDK2 P24941 1/20 0.50
IKBKE Q14164 1/20 0.50
PIK3CG P48736 1/20 0.46
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4398692 0.93 PLK1 (0.66) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4413899 0.84 PLK1 (0.62) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4632568 0.82 PLK1 (0.59) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4406541 0.82 PLK1 (0.69) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4397740 0.81 PLK1 (0.55) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL2980041 0.79 PLK1 (0.72) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4404339 0.79 PLK1 (0.72) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4400238 0.79 PLK1 (0.72) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL4404140 0.79 PLK1 (0.61) PLK1PLK3NEK2PIK3CDNUAK1
SCHEMBL14029456 0.79 PLK1 (0.65) PLK1PLK3NEK2PIK3CDNUAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924572-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SmithKline Beecham Corporation (US) 2008-05-28 EP disclosed
WO-2007030366-A1 REGIOSELECTIVE PROCESS FOR PREPARING BENZIMIDAZOLE THIOPHENES SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed