SCHEMBL4632610

SCHEMBL4632610

CC(C)CCc1ccc(CBr)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
TRPA1 O75762 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
AOC3 Q16853 2/20 0.34
OPRK1 P41145 5/20 0.34
OPRM1 P35372 4/20 0.34
OPRD1 P41143 4/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ADRB2 P07550 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8080450 0.87 HTT (0.41) TSHRHTTSMN1; SMN2AOC3OPRK1
SCHEMBL30124796 0.82 HRH3 (0.42) TSHRTRPA1ALDH1A1OPRK1OPRM1
SCHEMBL6768070 0.81 TAAR1 (0.50) AOC3
SCHEMBL3047188 0.78 CYP1A2 (0.52) ALDH1A1
SCHEMBL31277039 0.78 TAAR1 (0.52) TSHRALDH1A1HTTSMN1; SMN2
SCHEMBL9045813 0.78 PTGS1 (0.45) TSHRALDH1A1
SCHEMBL7717163 0.77 TSHR (0.39) TSHRTRPA1ALDH1A1HTTSMN1; SMN2
SCHEMBL13260233 0.76 CYP1A2 (0.45)
SCHEMBL2741643 0.76 CHKA (0.41) TSHRHTTSMN1; SMN2OPRK1KDM4E
SCHEMBL22047479 0.76 HTT (0.35) TSHRHTTSMN1; SMN2AOC3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed