SCHEMBL4633215

SCHEMBL4633215

[2H]C([2H])(Nc1cc(C(=O)N(C)C)cc2c1nc(C)n2C([2H])([2H])[2H])c1c(C)cccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.41
CYP2C9 P11712 5/20 0.41
CYP1A2 P05177 5/20 0.41
CYP2C19 P33261 5/20 0.41
CYP2D6 P10635 3/20 0.41
CD38 P28907 3/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
KCNH2 Q12809 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
PABPC1 P11940 1/20 0.31
CASP1 P29466 1/20 0.31
HTT P42858 1/20 0.31
HSD17B10 Q99714 1/20 0.31
FYN P06241 1/20 0.31
PTK2 Q05397 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592754 0.84 CYP3A4 (0.61) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL4634189 0.83 CYP3A4 (0.50) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5902197 0.80 CYP3A4 (0.53) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5901943 0.79 CYP3A4 (0.52) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5901801 0.77 CYP3A4 (0.53) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL4592785 0.77 CYP3A4 (0.46) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5902100 0.77 CYP3A4 (0.48) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5901446 0.75 CYP3A4 (0.47) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL5901927 0.75 CYP3A4 (0.47) CYP3A4CYP2C9CYP1A2CYP2C19CYP2D6
SCHEMBL4633218 0.75 KDM4E (0.33) ALDH1A1HPGDKDM4EGAAPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP claimed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO claimed
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP disclosed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO disclosed