SCHEMBL4634398

SCHEMBL4634398

COC(=O)Cc1cc(Br)ccc1OCC(=O)N1CCC(C#N)(Cc2cccc(Cl)c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.41
ALDH1A1 P00352 3/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 5/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
PTGER1 P34995 1/20 0.38
KDM4E B2RXH2 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
HTT P42858 2/20 0.37
TSHR P16473 2/20 0.37
GAA P10253 2/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
CCR5 P51681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4634528 0.91 PTGDR2 (0.45) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL4633816 0.91 RECQL (0.43) RECQLALDH1A1HPGDNPSR1LMNA
SCHEMBL4634773 0.86 MAPK1 (0.41) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL4633988 0.84 RECQL (0.41) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL4634679 0.83 CCR1 (0.46) PTGDR2HPGDNPSR1LMNAPOLB
SCHEMBL4634685 0.82 RECQL (0.45) RECQLALDH1A1PTGDR2HPGDNPSR1
SCHEMBL4634364 0.77 PTGDR2 (0.43) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL5673235 0.76 RECQL (0.44) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL4634923 0.75 MAPK1 (0.49) RECQLALDH1A1PTGDR2PKMHPGD
SCHEMBL4633914 0.75 SMN1; SMN2 (0.38) ALDH1A1HPGDLMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928829-A1 PIPERIDINE DERIVATIVES AS ANTAGONISTS OF THE CC CHEMOKINE RECEPTOR CCR1 AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Schering Aktiengesellschaft (DE) 2008-06-11 EP claimed
WO-2006066948-A1 PIPERIDINE DERIVATIVES AS ANTAGONISTS OF THE CC CHEMOKINE RECEPTOR CCR1 AND THEIR USE AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2006-06-29 WO claimed