SCHEMBL4634512

SCHEMBL4634512

CO/C(=C1/SC(Nc2ccc(CC(=O)O)cc2)=NC1=O)c1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.51
PTGDR2 Q9Y5Y4 9/20 0.41
PDE4B Q07343 6/20 0.40
PDE4D Q08499 2/20 0.40
IKBKB O14920 1/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP7 Q9BQF6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4634520 1.00 NR1H4 (0.51) NR1H4PTGDR2PDE4BPDE4DIKBKB
SCHEMBL4120866 0.82 PTGS1 (0.48) NR1H4PDE4BPDE4D
SCHEMBL4120873 0.82 PTGS1 (0.48) NR1H4PDE4BPDE4D
Acetic Acid SCHEMBL4634751 0.79 CYP26A1 (0.37) NR1H4NPC1CASP3RAB9ASENP7
Acetic Acid SCHEMBL4634752 0.79 CYP26A1 (0.37) NR1H4NPC1CASP3RAB9ASENP7
Acetic Acid SCHEMBL4635060 0.78 DHODH (0.39) NPC1CASP3RAB9ASENP7
Acetic Acid SCHEMBL4635062 0.78 DHODH (0.39) NPC1CASP3RAB9ASENP7
Acetic Acid SCHEMBL4129774 0.78 CSNK2A2 (0.35) NPC1CASP3RAB9ASENP7
SCHEMBL4134807 0.76 NR1H4 (0.50) NR1H4PDE4BPDE4D
SCHEMBL4134811 0.76 NR1H4 (0.50) NR1H4PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934192-A1 THIAZOLINONES AND OXAZOLINONES AND THEIR USE AS PTP1B INHIBITORS Torrent Pharmaceuticals Ltd (IN) 2008-06-25 EP claimed
WO-2007032028-A1 THIAZOLINONES AND OXAZOLINONES AND THEIR USE AS PTP1B INHIBITORS TORRENT PHARMACEUTICALS LTD. (IN) 2007-03-22 WO claimed