SCHEMBL463573

SCHEMBL463573

[CH2]COOCC=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30185 0.86
SCHEMBL1576596 0.82
SCHEMBL170804 0.82
Hydrogen Peroxide SCHEMBL16402637 0.79 TSHR (0.38)
Butane SCHEMBL3845806 0.73 TSHR (0.42)
SCHEMBL181037 0.73
SCHEMBL1386758 0.72
SCHEMBL16402640 0.71 TSHR (0.32)
SCHEMBL367516 0.71
SCHEMBL2066 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130108858-A1 Methods for Making an Article Coated with a Photochromic Film and Use Thereof in Ophthalmological Optics Essilor International (Compagnie Generate d Optique (FR) 2013-05-02 US claimed
JP-2009525497-A 2009-07-09 JP claimed
US-20090169859-A1 Article Comprising a Mesoporous Coating Having a Refractive Index Profile and Methods for Making Same ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2009-07-02 US claimed
EP-1979281-A1 METHODS FOR MAKING AN ARTICLE COATED WITH A PHOTOCHROMIC FILM AND USE THEREOF IN OPHTHALMOLOGICAL OPTICS ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2008-10-15 EP claimed
EP-1979770-A2 ARTICLE COMPRISING A MESOPOROUS COATING HAVING A REFRACTIVE INDEX PROFILE AND METHODS FOR MAKING SAME ESSILOR INTERNATIONAL Compagnie Générale d'Optique (FR) 2008-10-15 EP claimed
WO-2007090983-A2 ARTICLE COMPRISING A MESOPOROUS COATING HAVING A REFRACTIVE INDEX PROFILE AND METHODS FOR MAKING SAME ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2007-08-16 WO claimed
WO-2007088312-A1 METHODS FOR MAKING AN ARTICLE COATED WITH A PHOTOCHROMIC FILM AND USE THEREOF IN OPHTHALMOLOGICAL OPTICS ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2007-08-09 WO claimed
EP-3172375-B1 FIBROUS SUPPORT COMPRISING PARTICLES CONTAINING A PARTIALLY WATER-SOLUBLE ACTIVE AGENT, PARTICLES, AND METHODS FOR PRODUCING SAID PARTICLES SATISLOH AG (CH) 2024-03-13 EP disclosed
EP-4235273-A2 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS Essilor International (FR) 2023-08-30 EP disclosed
EP-3027396-B1 ADDITIVE MANUFACTURING PROCESSES FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INT (FR) 2023-06-14 EP disclosed
EP-3172375-A1 FIBROUS SUPPORT COMPRISING PARTICLES CONTAINING A PARTIALLY WATER-SOLUBLE ACTIVE AGENT, PARTICLES, AND METHODS FOR PRODUCING SAID PARTICLES Satisloh AG (CH) 2017-05-31 EP disclosed
US-9534160-B2 Method for manufacturing a substrate coated with mesoporous antistatic film, and use thereof in ophthalmic optics ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2017-01-03 US disclosed
US-20160167299-A1 ADDITIVE MANUFACTURING FOR TRANSPARENT OPHTHALMIC LENS ESSILOR INTERNATIONAL (FR) 2016-06-16 US disclosed
US-20090169859-A1 Article Comprising a Mesoporous Coating Having a Refractive Index Profile and Methods for Making Same ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2009-07-02 US disclosed
EP-1979281-A1 METHODS FOR MAKING AN ARTICLE COATED WITH A PHOTOCHROMIC FILM AND USE THEREOF IN OPHTHALMOLOGICAL OPTICS ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2008-10-15 EP disclosed
EP-1979770-A2 ARTICLE COMPRISING A MESOPOROUS COATING HAVING A REFRACTIVE INDEX PROFILE AND METHODS FOR MAKING SAME ESSILOR INTERNATIONAL Compagnie Générale d'Optique (FR) 2008-10-15 EP disclosed
WO-2007090983-A2 ARTICLE COMPRISING A MESOPOROUS COATING HAVING A REFRACTIVE INDEX PROFILE AND METHODS FOR MAKING SAME ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2007-08-16 WO disclosed
WO-2007088312-A1 METHODS FOR MAKING AN ARTICLE COATED WITH A PHOTOCHROMIC FILM AND USE THEREOF IN OPHTHALMOLOGICAL OPTICS ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2007-08-09 WO disclosed
EP-1789508-A1 METHOD OF PRODUCING A SUBSTRATE WHICH IS COATED WITH A MESOPOROUS LAYER AND USE THEREOF IN OPHTHALMIC OPTICS ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2007-05-30 EP disclosed
WO-2006021698-A1 METHOD OF PRODUCING A SUBSTRATE WHICH IS COATED WITH A MESOPOROUS LAYER AND USE THEREOF IN OPHTHALMIC OPTICS ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 2006-03-02 WO disclosed