SCHEMBL4635999

SCHEMBL4635999

C#CCn1c(=O)c2c(nc(C#Cc3cccc(OC)c3)n2C)n(CCC=O)c1=O

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.55
ADORA2A P29274 2/20 0.55
ADORA2B P29275 1/20 0.55
GLA P06280 1/20 0.51
ADORA3 P0DMS8 1/20 0.45
MAOB P27338 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2539378 0.93 ADORA1 (0.56) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2538825 0.90 ADORA1 (0.53) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL8180993 0.89 ADORA1 (0.53) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2541029 0.89 ADORA1 (0.59) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2545534 0.89 ADORA1 (0.53) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2537627 0.89 ADORA1 (0.57) ADORA1ADORA2AADORA2BGLAMAOB
SCHEMBL2540207 0.89 ADORA1 (0.53) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2542723 0.88 ADORA1 (0.51) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2540252 0.88 ADORA1 (0.67) ADORA1ADORA2AADORA2BGLAADORA3
SCHEMBL2542178 0.85 ADORA1 (0.49) ADORA1ADORA2AADORA2BGLAADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed