SCHEMBL4636591

SCHEMBL4636591

C#CCn1c(=O)c2c(nc(C#Cc3cccc(OC)c3)n2CC2CCC2)n(C)c1=O

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.54
ADORA2A P29274 7/20 0.52
MAOB P27338 4/20 0.52
ADORA3 P0DMS8 1/20 0.44
ADORA2B P29275 3/20 0.43
DPP4 P27487 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2548492 0.90 ADORA1 (0.57) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL4635978 0.87 ADORA1 (0.55) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL2537627 0.86 ADORA1 (0.57) ADORA1ADORA2AMAOBADORA2B
SCHEMBL4947786 0.85 ADORA1 (0.53) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL4950417 0.85 ADORA1 (0.53) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL4725744 0.85 ADORA1 (0.53) ADORA1ADORA2AMAOBADORA2B
SCHEMBL4636251 0.85 ADORA1 (0.53) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL4636192 0.84 ADORA1 (0.56) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL4636568 0.84 ADORA1 (0.52) ADORA1ADORA2AMAOBADORA3ADORA2B
SCHEMBL16199476 0.82 ADORA1 (0.56) ADORA1ADORA2AMAOBADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed