SCHEMBL4637175

SCHEMBL4637175

CCC1(CCOc2cccc(CC(=O)OC)c2)CCN(c2nc3ccc(Cl)cc3s2)CC1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 20/20 0.66
PPARG P37231 15/20 0.66
PPARA Q07869 6/20 0.66
CYP2C9 P11712 3/20 0.57
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL334711 0.88 PPARD (0.85) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL10219908 0.82 PPARD (0.60) PPARDPPARGPPARACYP2C9
SCHEMBL334847 0.81 PPARD (0.60) PPARDPPARGPPARACYP2C9
SCHEMBL10220994 0.80 PPARD (0.85) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL4637591 0.80 PPARD (0.59) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL334547 0.80 PPARD (1.00) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL10221068 0.79 PPARD (0.84) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL333917 0.79 PPARD (0.62) PPARDPPARGPPARACYP2C9
SCHEMBL10219891 0.79 PPARD (0.64) PPARDPPARGPPARACYP2C9
SCHEMBL334394 0.79 PPARD (0.59) PPARDPPARGPPARACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939189-A1 DERIVATIVE HAVING PPAR AGONISTIC ACTIVITY SHIONOGI & CO., LTD. (JP) 2008-07-02 EP disclosed