SCHEMBL4637262

SCHEMBL4637262

C#CCn1c(=O)c2c(nc(C#Cc3ccc(OC)c(OC)c3)n2C)n(CCCOC(C)=O)c1=O

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.44
ADORA2A P29274 5/20 0.44
ADORA2B P29275 3/20 0.44
ADORA1 P30542 2/20 0.44
ADORA3 P0DMS8 4/20 0.39
HTR1A P08908 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAOB P27338 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12233616 0.95 ADORA2A (0.41) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4949293 0.91 GLA (0.47) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL2542706 0.89 ADORA2A (0.55) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4950588 0.88 ADORA2A (0.42) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL12233850 0.88 GLA (0.58) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4952861 0.87 ADORA2A (0.45) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4944961 0.87 ADORA2A (0.48) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4950606 0.87 ADORA2A (0.43) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL4951704 0.86 ADORA2A (0.44) GLAADORA2AADORA2BADORA1ADORA3
SCHEMBL12233757 0.86 ADORA2A (0.42) GLAADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed