SCHEMBL4637283

SCHEMBL4637283

CCOc1ccc(C(CC(=O)O)N2C(=O)c3ccccc3C2=O)cc1OC1CCCC1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 13/20 0.82
PDE4B Q07343 13/20 0.82
PDE4C Q08493 13/20 0.82
PDE4D Q08499 13/20 0.82
TNF P01375 8/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5905279 0.94 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4637184 0.91 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4637637 0.91 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4637167 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL5905326 0.90 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4637688 0.89 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL5905040 0.89 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL6692793 0.88 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL5905230 0.87 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DTNF
SCHEMBL4637202 0.86 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1468991-B1 Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORP (US) 2008-02-20 EP claimed
EP-1468991-A1 Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORPORATION (US) 2004-10-20 EP claimed
EP-1468991-B1 Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORP (US) 2008-02-20 EP disclosed
EP-1468991-A1 Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORPORATION (US) 2004-10-20 EP disclosed
EP-0874819-B1 IMIDES AS PDE III, PDE IV AND TNF INHIBITORS CELGENE CORP (US) 2004-05-26 EP disclosed
CN-1092640-C Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORP (US) 2002-10-16 CN disclosed
CN-1206405-A Imides as PDE III, PDE IV and TNF inhibitors CELGENE CORP (US) 1999-01-27 CN disclosed
EP-0874819-A1 IMIDES AS PDE III, PDE IV AND TNF INHIBITORS CELGENE CORPORATION (US) 1998-11-04 EP disclosed
US-5728844-A INHIBITORS OF TUMOR NECROSIS AND PHOSPHODIESTERASE CELGENE CORPORATION (US) 1998-03-17 US disclosed
WO-1997023457-A1 IMIDES AS PDE III, PDE IV AND TNF INHIBITORS CELGENE CORPORATION (US) 1997-07-03 WO disclosed