SCHEMBL4637336

SCHEMBL4637336

CCn1c(=O)c2c(nc(C#Cc3ccc(OC)c(OC)c3)n2C)n(CC)c1=O

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.60
ADORA1 P30542 3/20 0.60
ADORA3 P0DMS8 2/20 0.60
ADORA2B P29275 2/20 0.60
MAOB P27338 2/20 0.60
HTR1A P08908 1/20 0.60
CYP2C9 P11712 1/20 0.60
PDE4A P27815 1/20 0.60
PDE4D Q08499 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2535848 0.92 ADORA2A (0.52) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL14887293 0.91 ADORA2A (0.52) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL4952167 0.87 ADORA2A (0.54) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL12233689 0.87 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL14887294 0.87 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL4953221 0.86 ADORA2A (0.52) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL14887287 0.86 ADORA2A (0.51) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL4636181 0.85 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL16199497 0.84 ADORA2A (0.50) ADORA2AADORA1ADORA3ADORA2BMAOB
SCHEMBL4951282 0.83 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed