SCHEMBL4639258

SCHEMBL4639258

CCc1nnn(C2CC(n3cnc4c(NCC(c5ccccc5)c5ccccc5)nc(N5CCC(NC(=O)OC(C)(C)C)C5)nc43)C(O)C2O)n1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.42
ADORA3 P0DMS8 7/20 0.42
ADORA2B P29275 2/20 0.39
ADORA1 P30542 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2804736 1.00 ADORA2A (0.42) ADORA2AADORA3ADORA2BADORA1
SCHEMBL14289845 1.00 ADORA2A (0.42) ADORA2AADORA3ADORA2BADORA1
SCHEMBL2804739 1.00 ADORA2A (0.42) ADORA2AADORA3ADORA2BADORA1
SCHEMBL2804742 1.00 ADORA2A (0.42) ADORA2AADORA3ADORA2BADORA1
Trifluoroacetic Acid SCHEMBL589844 0.97 ADORA2A (0.41) ADORA2AADORA3ADORA2BADORA1
SCHEMBL589258 0.95 ADORA2A (0.38) ADORA2AADORA3ADORA2BADORA1
SCHEMBL589259 0.95 ADORA2A (0.38) ADORA2AADORA3ADORA2BADORA1
SCHEMBL589845 0.92 ADORA2A (0.38) ADORA2AADORA3ADORA2BADORA1
SCHEMBL10156338 0.92 ADORA2A (0.45) ADORA2AADORA3ADORA2BADORA1
SCHEMBL10155859 0.92 ADORA2A (0.45) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889846-A1 Purine derivatives as A2a agonists Novartis AG (CH) 2008-02-20 EP disclosed