SCHEMBL4654402

SCHEMBL4654402

CN(C)c1ncnc2ccc(-c3cccc(CN4C(=O)CCC4=O)c3)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 16/20 0.54
CLK4 Q9HAZ1 16/20 0.54
CYP3A4 P08684 15/20 0.54
LMNA P02545 11/20 0.54
ALDH1A1 P00352 10/20 0.54
MAPK1 P28482 9/20 0.54
TSHR P16473 9/20 0.54
USP2 O75604 5/20 0.54
CYP2D6 P10635 10/20 0.54
CYP2C19 P33261 9/20 0.54
HIF1A Q16665 5/20 0.54
GLA P06280 1/20 0.54
CYP2C9 P11712 4/20 0.52
HSD17B10 Q99714 4/20 0.51
MEN1 O00255 1/20 0.51
TP53 P04637 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
KMT2A Q03164 1/20 0.51
HPGD P15428 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4190916 0.99 CYP1A2 (0.53) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4177706 0.89 MAP4K4 (0.46) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4168730 0.87 MAP4K4 (0.43) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4187763 0.83 MAP4K4 (0.56) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4188366 0.82 CYP1A2 (0.56) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4654175 0.80 CD38 (0.47) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4178315 0.80 CYP3A4 (0.48) CYP1A2CLK4CYP3A4LMNAALDH1A1
Hydrochloric Acid SCHEMBL4182086 0.79 CD38 (0.46) CYP1A2CLK4CYP3A4LMNAALDH1A1
Hydrochloric Acid SCHEMBL4184206 0.79 CD38 (0.47) CYP1A2CLK4CYP3A4LMNAALDH1A1
SCHEMBL4176493 0.79 CLK4 (0.54) CYP1A2CLK4CYP3A4LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996562-A1 SUBSTITUTED 4-AMINO-QUINAZOLINE DERIVATIVES AS REGULATORS OF METABOTROPIC GLUTAMATE RECEPTORS AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-12-03 EP claimed
WO-2007104560-A1 SUBSTITUTED 4-AMINO-QUINAZOLINE DERIVATIVES AS REGULATORS OF METABOTROPIC GLUTAMATE RECEPTORS AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-09-20 WO claimed